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Etizolam 1 mg mikro pelete

Etizolam micro pellets properties

Sinonim 4-(2-klorofenil)-2-etil-9-metil-6H-tieno[3,2-f][1,2,4]triazolo[4,3-a][1,4]diazepin
CAS broj : 40054-69-1
Formula C17H15ClN4S
Molarna masa : 342,8 g/mol
Čistoća : ≥ 99%

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Etizolam 1 MG Micro Pellets – Precision Dosing for Research Purposes

Product Name: Etizolam 1 mg Micro Pellets
Active Substance: Etizolam
Chemical Class: Thienodiazepine (benzodiazepine analogue)
Molekularna formula: C17H15ClN4S
Molecular Mass: 342.85 g/mol
Form: Micro Pellets (submillimeter size)
Dosage: 1 mg per pellet
Pakiranje: 10 / 25 / 50 / 100 pellets
Application: For laboratory and analytical research only


🔬 What is Etizolam?

Etizolam is a thienodiazepine compound structurally related to traditional benzodiazepines. It is known for its potent GABA-A receptor agonism , which produces anxiolytic, sedative, and muscle relaxant effects . In analytical studies, Etizolam is being evaluated for its receptor binding profile , stability , and structural-activity relationships (SAR) within the benzodiazepine family.

The micro pellet shape offers exceptional precision dosing and reproducibility , ideal for fine-mesh laboratory applications and storage.


Primjene u istraživanju

  • Neuroreceptor analysis: GABA-A modulation in vitro
  • Structural activity study (SAR): Comparison with classical benzos (diazepam, alprazolam)
  • Stability studies: Under the influence of temperature, moisture and light
  • Pharmacokinetics (preclinical): In vivo simulations under ethical protocol
  • Analytical reference substance: LC-MS, HPLC, NMR

⚠️ Oprez: Not suitable for human or animal consumption. For professional research purposes only.


⚠️ Risks and Limitations

  • Very potent in low doses – incorrect use can be dangerous
  • Dependency potential with abuse
  • Possible regulation in EU/US – considered a controlled substance in some countries
  • Not intended for recreational use or self-experimentation
  • May cause drowsiness or motor disorders if handled incorrectly

🧪 Laboratory details

CharacteristicSpecification
Active substanceEtizolam (≥99% purity – HPLC, GC-MS)
FormMicro pellets (approximately 0.6–0.8 mm diameter)
Doziranje1 mg per pellet
ColourWhite to light gray
Stability≥ 24 months when stored correctly
SolubilitySoluble in ethanol, DMSO, acetonitrile
Savjeti za skladištenjeDark, dry, cool (2–8 °C)
Potvrda o autentičnostiAvailable upon request

💡 Recommended Use Cases

Research areaApplication
Studije vezanja receptoraGABA-A response in different subtypes
Analitička kemijaReference in HPLC or LC-MS equipment
Stability testingUnder stressful conditions in the laboratory
SAR researchComparison with other thienodiazepines

Često postavljana pitanja (FAQ)

1. What is the difference between a micro pellet and a regular pellet?
Micro pellets are much smaller (submillimeter size) and designed for highly accurate dosing and rapid dissolution during analytical processes.

2. Is Etizolam legal?
That varies by country. In some regions, Etizolam is a controlled substance . Always check the regulations in your country before ordering or using it.

3. Is this product suitable for human consumption?
No. These pellets are intended for laboratory use only . Use on humans or animals is prohibited and potentially dangerous.

4. How should I store the pellets?
Store them in a tightly closed, dry container at 2–8°C , protected from light and moisture.

5. Is a Certificate of Analysis available?
Yes, a COA (Potvrda o analizi) is available upon request for each batch. This includes HPLC data, purity, and lot number.


📦 Product overview

FeatureSpecification
Product nameEtizolam 1 mg mikro pelete
FormSubmillimeter pressed pellets
Doziranje1 mg per pellet
Pakiranje10 / 25 / 50 / 100 pellets
Čistoća≥99%
UsageFor laboratory use only
Storage conditionCool, dry, light-free
Legal statusRegion dependent
Potvrda o autentičnostiAvailable per batch

 

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